A - Human Necessities – 61 – K
Patent
A - Human Necessities
61
K
A61K 31/5375 (2006.01) C07D 207/04 (2006.01) C07D 413/02 (2006.01)
Patent
CA 2540061
The present invention is directed to certain phenyl pyrrolidine ether compounds which are useful as neurokinin-1 (NK-1) receptor antagonists, and inhibitors of tachykinin and in particular substance P. The invention is also concerned with pharmaceutical formulations comprising these compounds as active ingredients and the use of the compounds and their formulations in the treatment of certain disorders, including emesis, depression, and anxiety.
La présente invention concerne des composés à base de phényle pyrrolidine éther utilisés comme antagonistes du récepteur de la neurokinine-1 (NK-1) et des inhibiteurs de la tachykinine et plus particulièrement de la substance P. L'invention concerne également des préparations pharmaceutiques utilisant ces composés comme ingrédients actifs et l'application de ces compositions et de leurs préparations dans le traitement de certains troubles, y compris les vomissements, la dépression et l'anxiété.
Devita Robert J.
Lin Peter
Mills Sander G.
Young Jonathan R.
Merck & Co. Inc.
Norton Rose Or S.e.n.c.r.l. S.r.l./llp
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