Delivery of nucleic acid molecules to mucosal tissue

A - Human Necessities – 61 – K

Patent

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Details

A61K 48/00 (2006.01) A61K 31/70 (2006.01) A61K 39/21 (2006.01) A61K 39/29 (2006.01) C07K 14/02 (2006.01) C07K 14/15 (2006.01) C07K 14/16 (2006.01) C07K 14/18 (2006.01)

Patent

CA 2208524

Methods of introducing genetic material into cells of an individual are disclosed. Methods of inducing mucosal immunity in individuals against proteins and peptides are disclosed. The methods comprise the step of administering topically or by lavage into mucosal tissue selected from the group of mucosal tissue consisting of rectal, vaginal, urethral, sublingual and buccal, a nucleic acid molecule that comprises a nucleotide sequence that encodes a protein or peptide that comprises an epitope against which mucosal immunity is desired. The methods may be used to immunize an individual against a pathogen infection, hyperproliferative diseases or autoimmune diseases using nucleic acid molecules which encode proteins and peptides that share an epitope with a pathogen antigen or protein associated with cells involved in hyperproliferative diseases of autoimmune diseases, respectively. Methods of treating individuals are disclosed that comprise the step of administering topically or by lavage into mucosal tissue selected from the group consisting of rectal, vaginal, urethral, sublingual and buccal, a nucleic acid molecule that comprises a nucleotide sequence that encodes a therapeutic protein.

L'invention porte sur des procédés d'introduction de matériel génétique dans les cellules d'un individu et sur des procédés suscitant chez des individus l'immunité des muqueuses vis-à-vis de protéines et de peptides. Ces procédés consistent à administrer topiquement ou par lavage à un tissu muqueux (rectal, vaginal, urétral, sublingual ou buccal) une molécule d'acide nucléique comportant une séquence d'un nucléotide codant pour une protéine ou un peptide comportant un épitope contre lequel l'immunité de la muqueuse est souhaitée. Ces procédés peuvent servir pour immuniser des individus contre une infection pathogène, contre des maladies hyperprolifératives ou des maladies auto-immunes à l'aide de molécules d'acides nucléiques codant pour des protéines et des peptides qui partagent un épitope avec un antigène ou une protéine associés à des cellules impliquées dans des maladies hyperprolifératives ou auto-immunes. L'invention porte également sur des méthodes de traitement des individus consistant à administrer topiquement ou par lavage à un tissu muqueux (rectal, vaginal, urétral, sublingual ou buccal) une molécule d'acide nucléique comportant une séquence d'un nucléotide codant pour une protéine à effet thérapeutique.

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