C - Chemistry – Metallurgy – 07 – H
Patent
C - Chemistry, Metallurgy
07
H
C07H 19/23 (2006.01) A61K 31/7042 (2006.01) A61P 31/04 (2006.01) A61P 33/02 (2006.01) A61P 35/00 (2006.01) A61P 37/02 (2006.01)
Patent
CA 2514992
The present invention relates to a new process for the preparation of compounds of general formula (I) which are inhibitors of purine nucleoside phosphorylases (PNP), purine phosphoribosyltransferases (PPRT), 5'- methylthioadenosine phosphorylases (MTAP), 5'-methylthioadenosine nucleosidases (MTAN) and/or nucleoside hydrolases (NH).The present invention relates to a new process for the preparation of compounds of general formula (I) which are inhibitors of purine nucleoside phosphorylases (PNP), purine phosphoribosyltransferases (PPRT), 5'-methylthioadenosine phosphorylases (MTAP), 5'-methylthioadenosine nucleosidases (MTAN) and/or nucleoside hydrolases (NH).
La présente invention concerne un nouveau procédé de préparation de composés de formule générale (I) qui sont des inhibiteurs de purine nucléosides phosphorylases (PNP), de purines phosphoribosyltransférases (PPRT), de 5'-méthylthioadénosine phosphorylases (MTAP), de 5'-méthylthioadénosine nucléosidases (MTAN) et/ou de nucléosides hydrolases (NH). La présente invention concerne un nouveau procédé de préparation de composés de formule générale (I) qui sont des inhibiteurs de purine nucléosides phosphorylases (PNP), de purine phosphoribosyltransférases (PPRT), de 5'-méthylthioadénosine phosphorylases (MTAP), de 5'-méthylthioadénosine nucléosidases (MTAN) et/ou de nucléosides hydrolases (NH).
Evans Gary Brian
Tyler Peter Charles
Albert Einstein College Of Medicine Of Yeshiva University
Bereskin & Parr Llp/s.e.n.c.r.l.,s.r.l.
Industrial Research Limited
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