Novel 2-decarboxy-2-phosphinico prostaglandin f analogs

C - Chemistry – Metallurgy – 07 – F

Patent

Rate now

  [ 0.00 ] – not rated yet Voters 0   Comments 0

Details

C07F 9/30 (2006.01) A61K 31/662 (2006.01) A61P 19/08 (2006.01) A61P 27/06 (2006.01)

Patent

CA 2380326

The invention provides novel Prostaglandin F analogs. In particular, the present invention is directed to compounds having a structure according to formula (I) wherein R1, R z, X, Y, V, a, b, W, and Z are defined below. This invention also includes optical isomers, diastereomers and enantiomers of the formula, and pharmaceutically-acceptable salts, biohydrolyzable amides, esters, and imides thereof. The compounds of the present invention are useful for the treatment of a variety of diseases and conditions, such as bone disorders and glaucoma. Accordingly, the invention further provides pharmaceutical compositions comprising these compounds. The invention still further provides methods of treatment for bone disorders and glaucoma using these compounds or the compositions containing them.

La présente invention concerne de nouveaux analogues de prostaglandine F. En particulier, cette invention concerne des composés dont la structure est représentée par la formule (I) dans laquelle R1, R2, X, Y, V, a, b, W, et Z sont définis ci-dessous. En outre, cette invention comprend des isomères optiques, des diastéréoisomères et énantiomères de la formule, des sels acceptables sur le plan pharmaceutique, des amides biohydrolysables, des esters, et des imides de ceux-ci. Les composés de cette invention sont utilisés dans le traitement de maladies et d'états pathologiques variées, tels que les troubles osseux ou le glaucome. De même, cette invention concerne des compositions pharmaceutiques contenant ces composés. En outre, cette invention concerne des méthodes de traitement des troubles osseux et du glaucome utilisant ces composés ou les compositions qui les renferment.

LandOfFree

Say what you really think

Search LandOfFree.com for Canadian inventors and patents. Rate them and share your experience with other people.

Rating

Novel 2-decarboxy-2-phosphinico prostaglandin f analogs does not yet have a rating. At this time, there are no reviews or comments for this patent.

If you have personal experience with Novel 2-decarboxy-2-phosphinico prostaglandin f analogs, we encourage you to share that experience with our LandOfFree.com community. Your opinion is very important and Novel 2-decarboxy-2-phosphinico prostaglandin f analogs will most certainly appreciate the feedback.

Rate now

     

Profile ID: LFCA-PAI-O-1570578

  Search
All data on this website is collected from public sources. Our data reflects the most accurate information available at the time of publication.