C - Chemistry – Metallurgy – 07 – D
Patent
C - Chemistry, Metallurgy
07
D
C07D 413/04 (2006.01) A61K 31/381 (2006.01) A61K 31/4245 (2006.01) A61P 35/00 (2006.01) C07D 413/14 (2006.01)
Patent
CA 2641933
The present invention relates to compounds of formula (I), and pharmaceutically acceptable salts and tautomers thereof. Compounds of the present invention are inhibitors of histone deacetylase (HDAC) and are useful for treating cellular proliferative diseases, including cancer. They are also useful for treating neurodegenerative diseases, mental retardation, 10 schizophrenia, inflammatory diseases, restenosis, immune disorders, diabetes, cardiovascular disorders and asthma.
La présente invention a pour objet des composés de formule I, ainsi que des sels et des tautomères de qualité pharmaceutique desdits composés. Les composés selon la présente invention sont des inhibiteurs de l'histone désacétylase (HDAC) et peuvent être employés dans le traitement de maladies de prolifération cellulaire, y compris le cancer. Ils peuvent également être employés dans le traitement de maladies neurodégénératives, des retards mentaux, de la schizophrénie, de maladies inflammatoires, de la resténose, des troubles immuns, du diabète, des troubles cardio-vasculaires et de l'asthme.
Ferrigno Federica
Jones Philip
Muraglia Ester
Ontoria Ontoria Jesus Maria
Scarpelli Rita
Istituto Di Ricerche Di Biologia Molecolare P. Angeletti Spa
Ogilvy Renault Llp/s.e.n.c.r.l.,s.r.l.
LandOfFree
Thiophene and thiazole substituted trifluoroethanone... does not yet have a rating. At this time, there are no reviews or comments for this patent.
If you have personal experience with Thiophene and thiazole substituted trifluoroethanone..., we encourage you to share that experience with our LandOfFree.com community. Your opinion is very important and Thiophene and thiazole substituted trifluoroethanone... will most certainly appreciate the feedback.
Profile ID: LFCA-PAI-O-1593127