C - Chemistry – Metallurgy – 07 – D
Patent
C - Chemistry, Metallurgy
07
D
C07D 413/04 (2006.01) A61K 31/381 (2006.01) A61K 31/4245 (2006.01) A61P 37/06 (2006.01) C07D 333/22 (2006.01) C07D 333/40 (2006.01)
Patent
CA 2635047
The invention relates to thiophene derivatives of formula (I) / their preparation and their use as pharmaceutically active compounds. Said compounds particularly act as immunosuppressive agents wherein: A represents *-CO-CH=CH- , *-CO-CH2CH2-, *-CO-CH2-NH-, wherein the sterisks indicate the bond that is linked to the thiophene group of Formula (I) , and R1-R3 are as defined in the claims.
La présente invention concerne des dérivés de thiophène de formule (I, ainsi que leur préparation et leur utilisation en tant que composés pharmaceutiquement actifs. Lesdits composés agissent plus particulièrement comme des agents immunosuppresseurs, A représentant *-CO-CH=CH-, *-CO-CH2CH2-, *-CO-CH2-NH-, les astérisques indiquant la liaison avec le groupe thiophène de formule (I) et R1-R3 étant tels que définis dans les revendications.
Bolli Martin
Lehmann David
Mathys Boris
Mueller Claus
Nayler Oliver
Actelion Pharmaceuticals Ltd
Gowling Lafleur Henderson Llp
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