Novel aryl glycinamide derivatives, method of producing said...

Details Novel aryl glycinamide derivatives, method of producing said... Novel aryl glycinamide derivatives, method of producing said...

C - Chemistry, Metallurgy

07

D

C07D 295/15 (2006.01) A61K 31/445 (2006.01) A61K 31/495 (2006.01) A61K 31/535 (2006.01) A61K 31/55 (2006.01) C07D 211/46 (2006.01) C07D 211/58 (2006.01) C07D 213/74 (2006.01) C07D 221/14 (2006.01) C07D 223/12 (2006.01) C07D 239/42 (2006.01) C07D 241/08 (2006.01) C07D 243/08 (2006.01) C07D 295/145 (2006.01) C07D 295/185 (2006.01) C07D 295/30 (2006.01) C07D 317/60 (2006.01) C07D 401/14 (2006.01)

Patent

CA 2247257

The invention relates to new arylglycinamide derivatives of general formula I (see formula I) and the pharmaceutically acceptable salts thereof, wherein R1 and R2 together with the N to which they are bound form a ring of the formula (see formula II) in which R3, R4, R5, Ar, R6, R7, R8, R9, R10, R11, r, s, and t have the meanings given in the specification and the preparation and use thereof. The new compounds are valuable neurokinin (tachykinin) antagonists.

L'invention concerne de nouveaux dérivés d'arylglycinamide de formule (I) et leurs sels pharmaceutiquement acceptables, formule dans laquelle R<1> et R<2>, conjointement avec le N auquel ils sont liés, forment un composé cyclique des formules (a), (b), (c) ou (d) dans lesquelles R<3>, R<4>, R<5>, Ar, R<6>, R<7>, R<8>, R<9>, R<10>, R<11>, r, s et t ont les notations indiquées dans la description. L'invention concerne également la production et l'utilisation de ces nouveaux composés qui sont de précieux antagonistes de la neurokinine (tachykinine).

Affiliated with

Also associated with

Rating

Novel aryl glycinamide derivatives, method of producing said... does not yet have a rating. At this time, there are no reviews or comments for this patent.

If you have personal experience with Novel aryl glycinamide derivatives, method of producing said..., we encourage you to share that experience with our LandOfFree.com community. Your opinion is very important and Novel aryl glycinamide derivatives, method of producing said... will most certainly appreciate the feedback.

Rate now

Comments { 0 }

Profile ID: LFCA-PAI-O-1606627