C - Chemistry – Metallurgy – 07 – D
Patent
C - Chemistry, Metallurgy
07
D
C07D 487/04 (2006.01) A61K 31/4985 (2006.01) A61P 3/10 (2006.01)
Patent
CA 2417106
The present invention refers to chemical compounds of formula (I) as well as pharmaceutically usable salts, solvates and esters thereof, wherein R1 to R8 have the significance given in claim 1. They can be used in the form of pharmaceutical preparations for the treatment or prevention of disorders of the central nervous system, damage to the central nervous system, cardiovascular disorders, gastrointestinal disorders, diabetes insipidus, obesity and sleep apnoea.
La présente invention concerne des composés chimiques de la formule (1) ainsi que les sels, solvates et esters pharmaceutiquement utilisables de ces derniers, dans laquelle R?1¿ à R?8¿ sont tels que définis dans la revendication 1. Les composés de l'invention peuvent être utilisés sous la forme de préparations pharmaceutiques pour le traitement ou la prévention des troubles du système nerveux central, des lésions du système nerveux central, des troubles cardiovasculaires, des troubles gastro-intestinaux, de l'obésité et de l'apnée du sommeil.
Bentley Jonathan Mark
Hebeisen Paul
Mattei Patrizio
Muller Marc
Richter Hans
F. Hoffmann-La Roche Ag
Gowling Lafleur Henderson Llp
Vernalis Research Limited
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