Photoactivation of endogenous porphyrins for treatment of...

A - Human Necessities – 61 – N

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A61N 5/06 (2006.01) A61B 6/00 (2006.01) A61K 41/00 (2006.01) A61K 49/00 (2006.01)

Patent

CA 2206203

Porphyrins, particularly protoporphyrin IX, are elevated in psoriatic plaques as compared to normal skin and skin of patients with other dermatological diseases. Psoriatic plaques with elevated porphyrin levels may be detected by fluorescence and spectral analysis. Endogenous porphyrins in psoriatic plaques may be activated with visible light to treat psoriatic plaques having elevated porphyrin concentrations. Skin conditions may be optimized to increase the endogenous synthesis of porphyrins in psoriatic plaques. A topical formulation may be applied to psoriatic plaques to optimize skin conditions such as pH, iron concentration, temperature, hydration, calcium concentration, oxygenation, electrical conductivity and estrogen concentration for increased production of endogenous porphyrins.

Les plaques psoriasiques ont une concentration élevée en porphyrines, en particulier en protoporphyrine IX, comparativement à la peau normale et à la peau des patients souffrant d'autres affections cutanées. Il est possible de détecter les plaques psoriasiques à concentration élevée en porphyrine par fluorescence et par analyse spectrale. Les porphyrines endogènes présentes dans les plaques psoriasiques peuvent être activées par la lumière visible pour traiter les plaques psoriasiques à concentration élevée en porphyrines. On peut optimiser les caractéristiques de la peau afin d'accroître la synthèse endogène de porphyrines dans les plaques psoriasiques. On peut appliquer une formulation topique sur les plaques psoriasiques pour optimiser les caractéristiques de la peau, telles que le pH, la concentration en fer, la température, l'hydratation, la concentration en calcium, l'oxygénation, la conductivité électrique et la concentration en oestrogènes de manière à accroître la production de porphyrines endogènes.

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