A - Human Necessities – 61 – K
Patent
A - Human Necessities
61
K
A61K 38/04 (2006.01) A61K 51/08 (2006.01)
Patent
CA 2614615
The present invention is directed to compounds according to formula, (R2R3)-A1- c(A2-A3-A4-A5-A6-A7-A8-A9)-A10-R1, and pharmaceutically-acceptable salts thereof that act as ligands for one or more of the melanocortin receptors, to methods of using such compounds to treat mammals and to pharmaceutical compositions comprising said compounds.
La présente invention concerne des composés représentés par la formule (R2R3)-A1-c(A2-A3-A4-A5-A6-A7-A8-A9)-A10-R1, et des sels acceptables d'un point de vue pharmaceutique de ceux-ci, servant de ligands pour un ou plusieurs récepteurs de la mélanocortine, des méthodes d'utilisation desdits composés dans le traitement des mammifères, et des compositions pharmaceutiques contenant lesdits composés.
Dong Zheng Xin
Moreau Jacques-Pierre
Ipsen Pharma S.a.s
Smart & Biggar
Societe de Conseils de Recherches Et D'applications Scientifique
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