C - Chemistry – Metallurgy – 07 – C
Patent
C - Chemistry, Metallurgy
07
C
C07C 317/44 (2006.01) A61K 31/277 (2006.01) A61K 47/48 (2006.01) A61P 35/00 (2006.01)
Patent
CA 2659746
Compounds useful as antiproliferative agents, including, for example, anticancer agents, according to formula (I): wherein Ar1, Ar2, D, G, formula (a), m and n are as defined herein, salts, antibody conjugates, pharmaceutical compositions, methods of treatment, synthetic processes, and intermediates useful in such processes are provided.
L'invention concerne des composés utiles comme agents anti-prolifératifs, comprenant, par exemple, des agents anti-cancer, selon la formule (I) : dans laquelle Ar1, Ar2, D, G, la formule (II), m et n sont tels que définis ici. L'invention concerne également des sels, des conjugués d'anticorps, des compositions pharmaceutiques, des procédés de traitement, des procédés de synthèse et des intermédiaires utiles dans de tels procédés.
Reddy E. Premkumar
Reddy M. V. Ramana
Borden Ladner Gervais Llp
Temple University - Of The Commonwealth System Of Higher Educati
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