Substituted cyclic urea derivatives and the use thereof as...

Details Substituted cyclic urea derivatives and the use thereof as... Substituted cyclic urea derivatives and the use thereof as...

C - Chemistry, Metallurgy

07

D

C07D 233/36 (2006.01) A61K 31/4166 (2006.01) A61K 31/4184 (2006.01) A61K 31/513 (2006.01) C07D 233/42 (2006.01) C07D 235/26 (2006.01) C07D 235/28 (2006.01) C07D 239/10 (2006.01)

Patent

CA 2605144

The invention relates to substituted cyclic urea derivatives, wherein X represents O, S or N-C=N; m is 1 or 2; n is 1 or 2; p1 and p2 represent independently 0, 1, 2 or 3, and the sum of p1 and p2 is 0, 1, 2 or 3. The invention also relates to methods for producing said derivatives, to drugs containing these compounds and to the use of these compounds for producing drugs. The inventive drugs are especially useful for vanilloid receptor 1 (VR1/TRPV1) regulation, preferably for vanilloid receptor 1 (VR1/TRPV1) inhibition and/or vanilloid receptor 1 (VR1/TRPV1) stimulation.

L'invention concerne des dérivés d'urée cycliques substitués de formule (I), dans laquelle X représente O, S ou N-C=N, m vaut 1 ou 2, n vaut 1 ou 2 et p1 et p2 valent indépendamment l'un de l'autre respectivement 0, 1, 2 ou 3, la somme de p1 et p2 étant égale à 0, 1, 2 ou 3. L'invention concerne également des procédés pour la production de ces composés, des médicaments contenant ces composés et l'utilisation de ces composés pour produire des médicaments. Les médicaments selon l'invention conviennent notamment pour la régulation du récepteur vanilloïde 1 (VR1/TRPV1), de préférence pour l'inhibition du récepteur vanilloïde 1 (VR1/TRPV1) et/ou pour la stimulation du récepteur vanilloïde 1 (VR1/TRPV1).

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