C - Chemistry – Metallurgy – 07 – D
Patent
C - Chemistry, Metallurgy
07
D
C07D 239/50 (2006.01) A61K 31/506 (2006.01) A61P 11/06 (2006.01) A61P 29/00 (2006.01) A61P 37/00 (2006.01)
Patent
CA 2643838
Disclosed are compounds, which bind VLA-4. Certain of these compounds also inhibit leukocyte adhesion and. in particular, leukocyte adhesion mediated by VLA-4. Such compounds are useful in the treatment of inflammatory diseases in a human or animal subject such as asthma, Alzheimer's disease, atherosclerosis, AIDS dementia, diabetes inflammatory bowel disease, Crohn's disease, rheumatoid arthritis, tissue transplantation, tumor metastasis and myocardial ischemia. The compounds can also be, administered for the treatment of inflammatory brain diseases such as multiple sclerosis.
La présente invention concerne des composés qui se lient à VLA-4. Certains de ces composés inhibent également l'adhésion leucocytaire et notamment l'adhésion leucocytaire médiée par VLA-4. De tels composés sont utiles pour le traitement des maladies inflammatoires chez l'être humain ou l'animal telles que l'asthme, la maladie d'Alzheimer, l'athérosclérose, la démence du SIDA, le diabète, la maladie inflammatoire des intestins, la maladie de Crohn, la polyarthrite rhumatoïde, la greffe de tissus, les métastases tumorales et l'ischémie myocardique. Les composés peuvent également être administrés pour le traitement de maladies inflammatoires cérébrales telles que la sclérose en plaques.
Konradi Andrei W.
Semko Christopher
Smith Jenifer L.
Xu Ying-Zi
Elan Pharmaceuticals Inc.
Ridout & Maybee Llp
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