A - Human Necessities – 61 – K
Patent
A - Human Necessities
61
K
A61K 31/404 (2006.01) A61P 5/24 (2006.01) C07D 403/04 (2006.01)
Patent
CA 2573314
Pyrrole-oxindole derivatives useful as progesterone receptor antagonists, and methods for preparing the same, are provided. Pharmaceutical compositions containing these derivatives are described, as is the use thereof in contraception and hormone-related conditions.
La présente invention décrit des dérivés de pyrrole-oxindole utilisés comme antagonistes des récepteurs de la progestérone, ainsi que les méthodes permettant de synthétiser lesdits dérivés. La présente invention décrit également des préparations pharmaceutiques comprenant lesdits dérivés, ainsi que l'utilisation desdites préparations à des fins contraceptives ou pour traiter des affections d'origine hormonale.
Fensome Andrew
Grubb Gary Sondermann
Marella Michael Anthony
Mccomas Casey Cameron
Melenski Edward George
Torys Llp
Wyeth
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