C - Chemistry – Metallurgy – 07 – D
Patent
C - Chemistry, Metallurgy
07
D
C07D 239/91 (2006.01) A61K 31/517 (2006.01) A61P 25/00 (2006.01) C07D 401/12 (2006.01) C07D 403/12 (2006.01) C07D 405/12 (2006.01)
Patent
CA 2568835
The present invention provides compounds of formula (I), their use as PARP inhibitors as well as pharmaceutical compositions comprising said compounds of formula (I) wherein R1, R2, R3, L, X, Y and Z have defined meanings.
La présente invention concerne des composés représentés par la formule (I) et leur utilisation en tant qu'inhibiteurs de PARP, ainsi que des compositions pharmaceutiques renfermant lesdits composés de formule (I). Dans cette formule, R1, R2, R3, L, X, Y et Z sont définis comme spécifié dans le descriptif.
Guillemont Jerome Emile Georges
Kennis Ludo Edmond Josephine
Mertens Josephus Carolus
Somers Maria Victorina Francisca
Van Dun Jacobus Alphonsus Josephus
Gowling Lafleur Henderson Llp
Janssen Pharmaceutica N.v.
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