Tissue plasminogen activator-like protease

C - Chemistry – Metallurgy – 12 – N

Patent

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Details

C12N 15/55 (2006.01) C07H 21/04 (2006.01) C12N 9/64 (2006.01) C12N 15/63 (2006.01) A61K 38/00 (2006.01)

Patent

CA 2291482

The present invention relates to a novel t-PALP protein which is a member of the serine protease family. In particular, isolated nucleic acid molecules are provided encoding the human t-PALP protein. t-PALP polypeptides are also provided as are vectors, host cells and recombinant methods for producing the same. The invention further relates to screening methods for identifying agonists and antagonists of t-PALP activity. Also provided are diagnostic methods for detecting circulatory system-related disorders and therapeutic methods for treating circulatory system-related disorders.

La présente invention a trait à une nouvelle protéine, la protéase du type activateur tissulaire du plasminogène (t-PALP), qui fait partie de la famille "sérine protéase". L'invention concerne en particulier des molécules d'acides nucléiques isolées codant la protéine t-PALP humaine. L'invention concerne en outre les polypeptides t-PALP, ainsi que les vecteurs, les cellules hôtes et les procédés recombinants de production de la t-PALP. Par ailleurs, l'invention se rapporte à des procédés de criblage permettant d'identifier les agonistes et antagonistes de l'activité de la t-PALP. L'invention concerne enfin des procédés de diagnostic, permettant de déceler des troubles liés au système circulatoire, et des procédés thérapeutiques permettant de traiter lesdits troubles.

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