C - Chemistry – Metallurgy – 07 – D
Patent
C - Chemistry, Metallurgy
07
D
C07D 487/10 (2006.01) A61K 31/4747 (2006.01) A61P 3/06 (2006.01) A61P 25/02 (2006.01)
Patent
CA 2663504
Disclosed are compounds of the formula (I), wherein Z1 is -CH2- or ~C(O)-, R4 and R5 are carbon chains (and optionally, together can form a C2 bridge), u and v are independently an integer of 0-3 such that there sum is from 3 to 5, and R2 is heteroaryl, and R1 and R3 are as defined herein. Also disclosed are methods of treating pain, and methods of inhibiting the absorption of cholesterol using a compound of formula (I).
La présente invention concerne des composés de la formule (I), dans laquelle Z1 est -CH2- ou -C(O)-, R4 et R5 sont des chaînes carbonées (et en option, peuvent former ensemble un pont C2), u et v sont indépendamment un nombre entier de 0 à 3 tel que leur somme est comprise entre 3 et 5, et R2 est un hétéroaryle, et R1 et R3 sont tels que définis dans le présent document. La présente invention concerne également des procédés de traitement de la douleur, et des procédés d'inhibition de l'absorption du cholestérol à l'aide d'un composé de formule (I).
Burnett Duane A.
Mckittrick Brian
Norton Rose Or S.e.n.c.r.l. S.r.l./llp
Schering Corporation
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