1- [ (4- [benzoyl (methyl) amino] -3- (phenyl) butyl]...

Details 1- [ (4- [benzoyl (methyl) amino] -3- (phenyl) butyl]... 1- [ (4- [benzoyl (methyl) amino] -3- (phenyl) butyl]...

C - Chemistry, Metallurgy

07

D

C07D 401/04 (2006.01) A61K 31/4523 (2006.01) A61P 1/00 (2006.01)

Patent

CA 2652443

The present invention relates to new compounds of formula (I) wherein R1, R2 and X are as defined in the description, as well as salts and enantiomers thereof. The invention also relates to pharmaceutical compositions comprising said compounds, and to the use of said compounds in therapy, e.g. in the treatment of gastrointestinal disorders. The invention further relates to processes for the preparation of the compounds. The compounds are neurokinin (NK) receptor antagonists.

La présente invention concerne de nouveaux composés de formule (I), dans laquelle R1, R2 et X sont tels que définis dans la description, ainsi que des sels et des énantiomères de ceux-ci. L'invention concerne également des compositions pharmaceutiques comprenant ces composés, ainsi que l'utilisation desdits composés en thérapie, p. ex. en traitement de troubles gastro-intestinaux. L'invention concerne en outre des procédés de préparation de ces composés, qui sont des antagonistes des récepteurs de la neurokinine (NK).

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