C - Chemistry – Metallurgy – 07 – D
Patent
C - Chemistry, Metallurgy
07
D
C07D 211/90 (2006.01) A61K 31/4422 (2006.01) A61K 31/443 (2006.01) A61K 31/4436 (2006.01) A61P 9/04 (2006.01) C07D 405/06 (2006.01) C07D 409/06 (2006.01)
Patent
CA 2544763
The present invention provides certain substituted 1,4-dihydropyridine compounds, including pure enantiomeric forms and pharmaceutical formulations thereof These compounds provide for elevation of .alpha.-MyHC protein levels and .alpha.-MyHC mRNA levels, and most frequently these same compounds provide simultaneous lowering of .beta.-MyHC protein levels and .beta.-MyHC mRNA levels. Thus, these compounds may be used alone or in conjunction with other drugs to treat heart failure.
La présente invention concerne certains composés de 1,4-dihydropyridine substitués, y compris des formes énantiomères pures et des préparations pharmaceutiques de ces composés. Ces composés permettent d'augmenter les taux de protéine A-MyHC et d'ARNm A-MyHC, et, le plus souvent, ces composés permettent de réduire simultanément les taux de protéine B-MyHC et d'ARNm B-MyHC. Ainsi, ces composés peuvent être utilisés seuls ou conjointement avec d'autres médicaments pour traiter l'insuffisance cardiaque.
Melvin Larry
Schreiber Kathy
Bcf Llp
Myogen Inc.
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