1-aminoalkyl-1h-indoles useful as analgesics, anti-...

Details 1-aminoalkyl-1h-indoles useful as analgesics, anti-... 1-aminoalkyl-1h-indoles useful as analgesics, anti-...

C - Chemistry, Metallurgy

07

D

167/208, 260/279

C07D 209/04 (2006.01) C07D 209/08 (2006.01) C07D 209/12 (2006.01) C07D 209/14 (2006.01) C07D 209/30 (2006.01) C07D 401/06 (2006.01) C07D 401/10 (2006.01) C07D 403/06 (2006.01) C07D 403/10 (2006.01) C07D 405/06 (2006.01) C07D 409/06 (2006.01) C07D 413/06 (2006.01) C07D 521/00 (2006.01)

Patent

CA 1258069

ABSTRACT OF THE DISCLOSURE Disclosed are novel 1-aminoalkyl-1H-indoles of the formula: Image (Ia) (wherein: R2 is hydrogen, alkyl, chloro, optionally substitut- ed phenyl or optionally substituted benzyl; R3 is optionally substituted cyclohexyl, optionally substituted phenyl, optionally substituted styryl, biphenyl, optionally substituted naphthyl, thienyl, furyl, benzofuryl, benzothienyl, quinolyl or alkylpyrrolyl; R4 is hydrogen, alkyl, hydroxy, alkoxy or halo; Alk is optionally alkyl-substituted alkylene; and N=B is azido, optionally substituted amino or optionally substituted cyclic amino such as morpholinyl, thio- morpholinyl, piperidinyl, pyrrolidinyl, azetidinyl, piperazinyl, hexahydrodiazepinyl or the N=B N-oxide thereof), which have analgesic, anti-rheumatic and anti-inflammatory activities and are useful as medicine.

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