2-aminothiazole allosteric enhancers of a1 adenosine receptors

Details 2-aminothiazole allosteric enhancers of a1 adenosine receptors 2-aminothiazole allosteric enhancers of a1 adenosine receptors

C - Chemistry, Metallurgy

07

D

C07D 277/60 (2006.01) A61K 31/428 (2006.01) C07D 277/84 (2006.01)

Patent

CA 2471989

The present invention relates generally to a class of 2-aminothiazole derivatives which have recently been identified as allosteric enhancers of the A1 adenosine receptor. These compounds, and therapeutic compositions containing them, are useful for treating conditions in which activation of the A1 adenosine receptor would be beneficial, for example, those conditions in which stimulation of angiogenesis would improve blood flow to ischemic tissues.

La présente invention concerne une classe de dérivés de 2-aminothiazoles récemment identifiés comme activateurs allostériques du récepteur de l'adénosine A1. Ces composés et les compositions thérapeutiques les contenant permettent de traiter les états pour lesquels l'activation du récepteur de l'adénosine A1 serait bénéfique, par exemple, les états pour lesquels la stimulation de l'angiogénèse améliorerait le débit sanguin vers les tissus ischémiques.

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