3-aminopropyloxyphenyl derivatives their preparation and...

Details 3-aminopropyloxyphenyl derivatives their preparation and... 3-aminopropyloxyphenyl derivatives their preparation and...

C - Chemistry, Metallurgy

07

D

167/207, 260/253

C07D 209/04 (2006.01) C07D 231/56 (2006.01) C07D 307/68 (2006.01)

Patent

CA 1296727

ABSTRACT OF TEE DISCLOSURE Compounds of Formula I, Image I characterised in that R signifies optionally substituted heteroaryl-, heteroarylalkyl or heteroarylalkenyl, R1 signifies hydrogen or a substituent, R2 is hydroxy or a group -Z-(CH2)n-Y-R3 wherein R3 is hydrogen, alkyl, hydroxyalkyl, alkenyl, cycloalkyl, cycloalkylalkylene. hydroxy substituted cycloalkyl or cycloalkylalkylene, or optionally substituted aryl or aralkyl or aralkenyl moiety, and Y signifies oxygen or sulfur, and either Z is an oxygen atom and n is 2 or 3, or Z is a bond and n is 1, 2 or 3, A signifies alkylene or branched alkylene of 2 to 5 carbon atoms, W signifies a bond or imino, and X signifies a bond or imino, and their physiologically hydrolysable derivatives, in which at least one hydroxy group is in esterified form. The compounds exhibit beta adrenoceptor blocking activity. Process for the preparation of the compounds are also disclosed.

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