A - Human Necessities – 61 – K
Patent
A - Human Necessities
61
K
A61K 31/404 (2006.01) A61P 25/00 (2006.01) A61P 25/24 (2006.01)
Patent
CA 2577511
The present invention relates to methods for treating a patient suffering from diseases or disorders of the central nervous system associated with the disturbance of the human circadian clock that are ameliorated by inhibition of casein kinase I.epsilon. activity such as , for example, mood disorders including major depressive disorder, bipolar I disorder and bipolar II disorder, and sleep disorders including circadian rhythm sleep disorders such as, for example, shift work sleep disorder, jet lag syndrome, advanced sleep phase syndrome and delayed sleep phase syndrome, with 3-arylthioindole-2- carboxamides, 5-substituted-3-arylthioindole-2-carboxamides and related analogues.
La présente invention concerne des procédés pour traiter un patient souffrant de maladies ou de troubles du système nerveux central associé(e)s à des troubles de l~horloge circadienne et qui sont amélioré(e)s par l~inhibition de l~activité de la caséine kinase I.epsilon., tel(le)s que, par exemple, les troubles de l~humeur y compris les troubles dépressifs majeurs, la psychose maniaco-dépressive I et la psychose maniaco-dépressive II, et les troubles du sommeil y compris les troubles du sommeil liés au rythme circadien tels que, par exemple, les troubles du sommeil liés au travail par équipes, les symptômes du décalage horaire, le syndrome d~avance de phase et le syndrome de retard de phase, avec les 3-arylthioindole-2-carboxamides, les 3-arylthioindole-2-carboxamides substitués en position 5, et les analogues apparentés.
Aventis Pharmaceuticals Inc.
Bereskin & Parr Llp/s.e.n.c.r.l.,s.r.l.
LandOfFree
3-arylthioindole-2-carboxamide derivatives and analogs... does not yet have a rating. At this time, there are no reviews or comments for this patent.
If you have personal experience with 3-arylthioindole-2-carboxamide derivatives and analogs..., we encourage you to share that experience with our LandOfFree.com community. Your opinion is very important and 3-arylthioindole-2-carboxamide derivatives and analogs... will most certainly appreciate the feedback.
Profile ID: LFCA-PAI-O-2004617