C - Chemistry – Metallurgy – 07 – D
Patent
C - Chemistry, Metallurgy
07
D
C07D 409/06 (2006.01) A61K 31/4535 (2006.01) A61P 11/06 (2006.01)
Patent
CA 2560649
The present invention extends to the compound of formula I, or a prodrug, pharmaceutically acceptable salt, or solvate of said compound. Furthermore, the present invention is directed to a pharmaceutical composition comprising a pharmaceutically effective amount of the compound of formula I, and a pharmaceutically acceptable carrier. Furthermore, the present invention is directed to the use of a compound of formula I as an inhibitor of tryptase, comprising introducing the compound into a composition comprising tryptase. In addition, the present invention is directed to the use of a compound of formula I for treating a patient suffering from, or subject to, a physiological condition in need of amelioration of an inhibitor of tryptase comprising administering to the patient a therapeutically effective amount of the compound of Claim 1. The present invention is directed also to the preparation of a compound of formula I.
Un composé de formule (I), ou un promédicament, un sel pharmaceutiquement acceptable ou un solvate dudit composé. Une composition pharmaceutique comprenant une quantité pharmaceutiquement efficace du composé de formule (I) et un support pharmaceutiquement acceptable. L'utilisation du composé de formule (I) comme inhibiteur de la tryptase consistant à introduire le composé dans une composition comprenant de la tryptase. Par ailleurs, on prévoit l'utilisation d'un composé de formule (I) pour le traitement d'un patient souffrant d'une pathologie physiologique nécessitant l'amélioration d'un inhibiteur de la tryptase consistant à administrer au patient une quantité thérapeutiquement efficace du composé. On prévoit en outre la préparation d'un composé de formule (I).
Czekaj Mark
Davis Larry
Gao Zhongli
Haddad El-Bdaoui
Levell Julian
Aventis Pharmaceuticals Inc.
Bereskin & Parr Llp/s.e.n.c.r.l.,s.r.l.
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