4,5-dihydro- (1h)-pyrazole derivatives as cannabinoid cb1...

Details 4,5-dihydro- (1h)-pyrazole derivatives as cannabinoid cb1... 4,5-dihydro- (1h)-pyrazole derivatives as cannabinoid cb1...

C - Chemistry, Metallurgy

07

D

C07D 231/06 (2006.01) A61K 31/40 (2006.01) A61P 25/00 (2006.01) C07C 49/213 (2006.01) C07D 403/12 (2006.01) C07D 405/06 (2006.01) C07D 409/04 (2006.01) C07D 409/06 (2006.01)

Patent

CA 2632582

This invention is directed to 4,5-dihydro -(1 H)-pyrazole (pyrazoline) derivatives as cannabinoid CB1 receptor modulators, to pharmaceutical compositions containing these compounds, to methods for the preparation of these compounds, methods for preparing novel intermediates useful for their synthesis, and methods for preparing compositions. The invention also relates to the uses of such compounds and compositions, particularly their use in administering them to patients to achieve a therapeutic effect in disorders in which CB1 receptors are involved, or that can be treated via manipulation of those receptors. The compounds have the general formula (I) wherein the symbols have the meanings given in the specification.

Cette invention concerne des dérivés de 4,5-dihydro-(1 H)-pyrazole (pyrazoline) en tant que modulateurs du récepteur cannabinoïde CB1, des compositions pharmaceutiques contenant ces composés, des procédés de fabrication de ces composés, des procédés de fabrication de nouveaux intermédiaires utiles pour leur synthèse et des procédés de préparation des compositions. L~invention concerne également l~utilisation de tels composés et de telles compositions, notamment leur utilisation pour une administration à des patients dans un but thérapeutique pour des troubles impliquant les récepteurs CB1 ou pouvant être traités par manipulation de ces récepteurs. Les composés ont la formule générale (I) dans laquelle les symboles ont les significations données dans la description.

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