4,5-dihydro-1h-pyrazole derivatives having cb1-antagonistic...

Details 4,5-dihydro-1h-pyrazole derivatives having cb1-antagonistic... 4,5-dihydro-1h-pyrazole derivatives having cb1-antagonistic...

C - Chemistry, Metallurgy

07

D

C07D 401/12 (2006.01) A61K 31/415 (2006.01) A61K 31/4155 (2006.01) A61K 31/454 (2006.01) A61K 31/4725 (2006.01) A61K 31/496 (2006.01) A61P 25/00 (2006.01) C07D 231/06 (2006.01) C07D 401/06 (2006.01) C07D 403/12 (2006.01) C07D 409/04 (2006.01)

Patent

CA 2456606

The present invention relates to a group of novel 4,5-dihydro-1H-pyrazole derivatives which are potent cannabinoid (CB1) receptor antagonists with utility for the treatment of diseases connected with disorders of the cannabinoid system. The compounds have the general formula (I) wherein the symbols have the meanings given in the specification. The invention also relates to methods for the preparation of these compounds, and to pharmaceutical compositions containing one or more of these compounds as an active component.

La présente invention concerne un groupe de nouveaux dérivés 4,5-dihydro-1H-pyrazole étant des antagonistes efficaces des récepteurs aux cannabinoïdes (CB1), et servant au traitement de troubles liés au système cannabinoïde. Les composés selon l'invention portent la formule générale (I) dans laquelle les symboles ont la signification donnée dans le descriptif. L'invention concerne également des procédés de fabrication desdits composés, ainsi que des compositions pharmaceutiques contenant un ou plusieurs de ces composés en tant qu'agent actif.

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