4,5-dihydro-1h-pyrazole derivatives having potent...

Details 4,5-dihydro-1h-pyrazole derivatives having potent... 4,5-dihydro-1h-pyrazole derivatives having potent...

C - Chemistry, Metallurgy

07

D

C07D 231/06 (2006.01) A61K 31/415 (2006.01) A61K 31/4155 (2006.01) A61K 31/4725 (2006.01) C07D 401/04 (2006.01) C07D 401/12 (2006.01) C07D 409/04 (2006.01)

Patent

CA 2442245

The present invention relates to a group of novel 4,5-dihydro-1H-pyrazole derivatives which are potent cannabinoid (CB1) receptor antagonists with utility for the treatment of diseases connected with disorders of the cannabinoid system. The compounds have the general formula (Ia) or (Ib) wherein the symbols have the meanings given in the specification. The invention also relates to methods for the preparation of these compounds, and to pharmaceutical compositions containing one or more of these compounds as an active component.

L'invention concerne un groupe de nouveaux dérivés 4,5-dihydro-1H-pyrazole qui sont de puissants antagonistes du récepteur (CB¿1?) des cannabinoïdes, utiles dans le traitement de maladies associées à des troubles du système cannabinoïde, ces composés étant représentés par la formule (Ia) ou (Ib) dans laquelle les symboles ont la signification indiquée dans la description. L'invention concerne également des procédés de préparation desdits composés et de compositions pharmaceutiques comprenant un ou plusieurs de ces composés utilisés en tant que composant actif.

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