4-aminotetrahydrobenzisoxazole or -isothiazole compounds

Details 4-aminotetrahydrobenzisoxazole or -isothiazole compounds 4-aminotetrahydrobenzisoxazole or -isothiazole compounds

C - Chemistry, Metallurgy

07

D

C07D 417/14 (2006.01) A61K 31/42 (2006.01) A61K 31/425 (2006.01) A61K 31/44 (2006.01) A61K 31/505 (2006.01) C07D 261/20 (2006.01) C07D 275/04 (2006.01) C07D 413/12 (2006.01) C07D 413/14 (2006.01) C07D 417/12 (2006.01)

Patent

CA 2213127

4-aminotetrahydrobenzisoxazole or -isothiazole compounds having general formulae (Ia) and (Ib), wherein R1-R6, X and P are further defined in the description. The disclosed compounds have GABA (4-aminobutanoic acid) inhibiting activity and are useful in the treatment of analgesia, psychosis, convulsions, anxiety or muscular and movement disorders, especially epilepsy.

Cette invention concerne des composés 4-aminotétrahydrobenzisoxazole ou -isothiazole représentés par les formules générales (Ia) et (Ib) dans lesquelles R?1¿-R?6¿, X et P sont définis par ailleurs dans le descriptif de l'invention. Ces composés présentent une activité inhibante vis-à-vis du GABA (acide 4-aminobutanoïque) et s'avèrent utiles pour le traitement de l'analgésie, de la psychose, des convulsions, de l'anxiété ou des troubles musculaires et des dyskinésies, et tout particulièrement de l'épilepsie.

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