C - Chemistry – Metallurgy – 07 – D
Patent
C - Chemistry, Metallurgy
07
D
C07D 309/32 (2006.01) A61K 31/365 (2006.01) A61K 31/38 (2006.01) A61K 31/415 (2006.01) A61K 31/44 (2006.01) C07C 323/22 (2006.01) C07D 211/86 (2006.01) C07D 311/96 (2006.01) C07D 335/02 (2006.01) C07D 405/02 (2006.01) C07D 405/04 (2006.01) C07D 405/12 (2006.01) C07D 407/06 (2006.01) C07D 409/04 (2006.01)
Patent
CA 2176043
The present invention relates to novel 5,6-dihydropyrone derivatives and related structures which potently inhibit the HIV aspartyl protease blocking HIV infectivity. The 5,6-dihydropyrone derivatives are useful in the development of therapies for the treatment of bacterial and viral infections amd diseases, including AIDS. The present invention is also directed to methods of synthesis of multifunctionalized 5,6-dihydroporones and of related structures.
La présente invention se rapporte à des nouveaux dérivés de la 5,6-dihydropyrone ainsi qu'à des structures apparentées, qui inhibent puissamment l'aspartyle protéase du VIH en bloquant le pouvoir infectant du VIH. Les dérivés de la 5,6-dihydropyrone sont utiles dans le développement des thérapies destinées au traitement des infections et maladies bactériennes et virales, notamment le SIDA. La présente invention se rapporte également à des procédés de synthèse des 5,6-dihydropyrones multifonctionnalisées et de structures apparentées.
Ellsworth Edmund Lee
Lunney Elizabeth
Tait Bradley Dean
Macrae & Co.
Warner-Lambert Company
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