6-h-pyrimido- (1,2-c) (1,3,5) benzoxadiazepines

Details 6-h-pyrimido- (1,2-c) (1,3,5) benzoxadiazepines 6-h-pyrimido- (1,2-c) (1,3,5) benzoxadiazepines

C - Chemistry, Metallurgy

07

D

260/238.5, 260/2

C07D 498/04 (2006.01) C07D 239/42 (2006.01)

Patent

CA 1051427

Abstract This invention relates to compounds of the formula Image X wherein m is 1 or 2; when m is 1, R occupies either position-4 or -5 of the starting 2-aminopyrimidine, but when R is halogen it occupies only position-5, when m is 2, the two R's occupy the 4- and 5-positions of the starting 2-aminopyrimidine, but only one of the two R-substituents can be halogen and it must occupy the 5-position; T is the same or different and is hydrogen, F, Cl, Br, alkyl of from 1 to 4 carbons, benzyl, phenyl, or mono-substituted phenyl wherein the substituent is F, Cl, Br, I, alkyl of from 1 to 4 carbons, alkoxy of from 1 to 4 carbons, or trifluoromethyl; R' is hydrogen, F, Cl, Br, I, alkyl of from 1 to 4 carbons, alkylsulfonyl wherein the alkyl radical has from 1 to 4 carbons, dialkylamidosulfonyl wherein each alkyl radical has from 1 to 4 carbons, trifluoro- methyl; n is 0 or 1; and R" is hydrogen or alkyl of from 1 to 4 carbons; and pharmaceutically acceptable acid-addition salts thereof, a process for preparing them and to intermediates therefor. These compounds exhibit central nervous system stimulating properties and act as muscle relaxants.

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