C - Chemistry – Metallurgy – 07 – D
Patent
C - Chemistry, Metallurgy
07
D
C07D 403/06 (2006.01) A61K 31/495 (2006.01) A61P 25/28 (2006.01) C07D 209/86 (2006.01) C07D 209/88 (2006.01) C07D 407/14 (2006.01) C07D 417/14 (2006.01)
Patent
CA 2385456
The present invention is related to piperazine derivatives of carbazole of formula (I) notably for use as pharmaceutically active compounds, as well as to pharmaceutical formulations containing such piperazine derivatives of carbazole. Said piperazine derivatives of carbazole are efficient modulators, in particular efficient inhibitors, of the Bax function and/or activation. The present invention is furthermore related to novel piperazine derivatives of carbazole as well as methods of their preparation.
La présente invention concerne des dérivés pipérazine de carbazole de formule (I) et plus spécifiquement l'utilisation de ces derniers en tant que composés pharmaceutiquement actifs ainsi que des formulations pharmaceutiques contenant de tels dérivés pipérazine de carbazole. Les dérivés pipérazine de carbazole sont des modulateurs efficaces, et plus particulièrement des inhibiteurs efficaces de la fonction et/ou de l'activation de Bax. Cette invention concerne également de nouveaux dérivés pipérazine de carbazole ainsi que des procédés de préparation de ces derniers.
Antonsson Bruno
Bombrun Agnes
Church Dennis
Gerber Patrick
Halazy Serge
Applied Research Systems Ars Holding N.v.
Kirby Eades Gale Baker
Merck Serono Sa
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