A - Human Necessities – 61 – K
Patent
A - Human Necessities
61
K
A61K 31/445 (2006.01) A61K 31/454 (2006.01) A61K 31/4545 (2006.01) C07D 413/14 (2006.01) C07D 417/14 (2006.01)
Patent
CA 2574156
Certain novel N-acylated piperidine derivatives are agonists of the human melanocortin receptor(s) and, in particular, are selective agonists of the human melanocortin-4 receptor (MC-4R). They are therefore useful for the treatment, control, or prevention of diseases and disorders responsive to the activation of MC-4R, such as obesity, diabetes, sexual dysfunction, including erectile dysfunction and female sexual dysfunction.
L'invention concerne certains nouveaux dérivés de pipéridine acylés qui sont des agonistes des récepteurs humains de la mélanocortine et, en particulier, des agonistes sélectifs du récepteur humain de la mélanocortine 4 (MC-4R). Ces dérivés s'avèrent ainsi utiles pour le traitement, la prévention de maladies et de troubles associés à l'activation du MC-4R et pour la lutte contre ces maladies et troubles, par exemple l'obésité, le diabète, les troubles de la sexualité, notamment les troubles de l'érection et les troubles de la sexualité chez la femme.
Bakshi Raman K.
Dellureficio James P.
Nargund Ravi P.
Merck & Co. Inc.
Merck Sharp & Dohme Corp.
Norton Rose Or S.e.n.c.r.l. S.r.l./llp
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