C - Chemistry – Metallurgy – 07 – D
Patent
C - Chemistry, Metallurgy
07
D
C07D 413/14 (2006.01) A61K 31/435 (2006.01) A61K 31/445 (2006.01) A61K 31/454 (2006.01) A61K 31/4545 (2006.01) A61K 31/47 (2006.01) A61K 31/495 (2006.01) A61K 31/55 (2006.01) C07D 211/62 (2006.01) C07D 211/64 (2006.01) C07D 211/68 (2006.01) C07D 217/02 (2006.01) C07D 223/16 (2006.01) C07D 401/06 (2006.01) C07D 401/12 (2006.01) C07D 401/14 (2006.01) C07D 403/06 (2006.01) C07D 413/06 (2006.01) C07D 491/08 (2006.01)
Patent
CA 2439149
Certain novel 4-substituted N-acylated piperidine derivatives are agonists of the human melanocortin receptor(s) and, in particular, are selective agonists of the human melanocortin-4 receptor (MC-4R). They are therefore useful for the treatment, control, or prevention of diseases and disorders responsive to the activation of MC-4R, such as obesity, diabetes, sexual dysfunction, including erectile dysfunction and female sexual dysfunction.
L'invention concerne certains nouveaux dérivés de pipéridine N-acétylée substitués en 4 utilisés comme agonistes du ou des récepteur(s) humain(s) de mélanocortine, et en particulier des agonistes sélectifs du récepteur humain de mélanocortine-4 (MC-4R). Ces dérivés sont utilisés pour traiter, lutter contre, ou prévenir des maladies et des troubles sensibles à l'activation de MC-4R, tels que l'obésité, les diabètes, un dysfonctionnement sexuel, notamment une dysfonction érectile et une dysfonction sexuelle chez la femme.
Bakshi Raman K.
Goulet Mark T.
Nargund Ravi P.
Sebhat Iyassu K.
Ujjainwalla Feroze
Merck & Co. Inc.
Merck Sharp & Dohme Corp.
Norton Rose Or S.e.n.c.r.l. S.r.l./llp
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