Alpha-(aryl-or heteroaryl-methyl)-beta piperidino...

C - Chemistry – Metallurgy – 07 – D

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C07D 451/06 (2006.01) A61K 31/46 (2006.01) A61P 25/04 (2006.01)

Patent

CA 2612299

This invention provides the compounds of formula (I), or a pharmaceutically acceptable salt thereof, wherein R1 and R2 independently represent hydrogen or the like; R3 and R4 independently represents hydrogen or the like; R5 represents aryl or the like; -X-Y- represents -CH2O- or the like; and n represents 0, 1 or 2.These compounds have ORL1 -receptor antagonist activity; and therefore, are useful to treat diseases or conditions such as pain, various CNS diseases etc.

La présente invention concerne les composés représentés par la formule (I) ou un sel pharmaceutiquement acceptable de ces derniers. Dans la formule, R1 et R2 représentent indépendamment hydrogène ou similaire; R3 et R4 représentent indépendamment hydrogène ou similaire; R5 représente aryle ou similaire; -X-Y- représente -CH2O- ou similaire; et n représente 0, 1 ou 2. Ces composés présentent une activité antagoniste du récepteur ORL1 et sont donc utiles pour traiter les maladies ou les pathologies telles que la douleur, diverses maladies du système nerveux central et autres. Formule (I)

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