Aminocyclopentanes and their preparation and pharmaceutical...

Details Aminocyclopentanes and their preparation and pharmaceutical... Aminocyclopentanes and their preparation and pharmaceutical...

C - Chemistry, Metallurgy

07

D

260/247.1, 260/2

C07D 295/14 (2006.01) C07C 405/00 (2006.01) C07D 295/096 (2006.01) C07D 295/112 (2006.01) C07D 295/155 (2006.01) C07D 333/16 (2006.01) C07D 409/12 (2006.01) C07D 521/00 (2006.01) C07F 7/18 (2006.01)

Patent

CA 1234811

ABSTRACT AMINOCYCLOPENTANES AND THEIR PREPARATION AND PHARMACEUTICAL FORMULATION Compounds are described of the formulae (1a) and (1b) Image in which: R1 is -H, C1-6 alkyl or C7-10 aralkyl, W is C1-7 alkylene X is cis or trans -CH=CH-, Y is a saturated heterocyclic amino group having 5-8 ring members, R2 is (i) substituted or unsubstituted phenylalkyl, thienylalkyl or naphthylalkyl or (ii) cinnamyl, and Z is -CH20H, -CHO or -CONHR4 where R4 is -H or methyl, and their salts and solvates. These compounds inhibit blood platelet aggregation, bronchoconstriction and vasoconstriction, and may be formulated for use as antithrombotic and antiasthmatic agents.

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