Analogs of .beta..sub.h-endorphin and process for the...

Details Analogs of .beta..sub.h-endorphin and process for the... Analogs of .beta..sub.h-endorphin and process for the...

C - Chemistry, Metallurgy

07

K

530/7.44

C07K 14/675 (2006.01) A61K 38/00 (2006.01)

Patent

CA 1102312

ABSTRACT A process for the preparation of .beta.h-endorphin analogs of the formula [X, Phe27, Gly21]-.beta.h-endorphin wherein X is null, Ala6,7, Nle5 or D-Thr2 and of physiologically acceptable acid addition salts thereof, characterized in that in the last step of a conventional solid or liquid phase synthesis the solid resin support and/or protecting groups of the protec- ted .beta.h-endorphin analogs are cleaved off in a manner know per se and that, if desired, physiologically acceptable acid addition salts are formed. The novel compounds exhibit analgesic activity.

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