Aqueous gel formulations containing immune reponse modifiers

A - Human Necessities – 61 – K

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Details

A61K 31/4745 (2006.01) A61K 31/20 (2006.01)

Patent

CA 2597092

Aqueous gel formulations, including an immune response modifier (IRM), such as those chosen from imidazoquinoline amines, tetrahydroimidazoquinoline amines, imidazopyridine amines, 6,7-fused cycloalkylimidazopyridine amines, 1,2 - bridged imidazoquinoline amines, imidazonaphthyridine amines, imidazotetrahydronaphthyridine amines, oxazoloquinoline amines, thiazoloquinoline amines, oxazolopyridine amines, thiazolopyridine amines, oxazolonaphthyridine amines, thiazolonaphthyridine amines, pyrazolopyridine amines, pyrazoloquinoline amines, tetrahydropyrazoloquinoline amines, pyrazolonaphthyridine amines, tetrahydropyrazolonaphthyridine amines, and lH- imidazo dimers fused to pyridine amines, quinoline amines, tetrahydroquinoline amines, naphthyridine amines, or tetrahydronaphthyridine amines, are provided. Methods of use and kits are also provided.

L'invention concerne des formulations de gel aqueux comprenant un modificateur de réponse immunitaire (IRM), tel que ceux choisis parmi les imidazoquinoline amines, les tétrahydroimidazoquinoline amines, les imidazopyridine amines, les cycloalkylimidazopyridine amines fusionnées en 6,7, les imidazoquinoline amines pontées en 1,2, les imidazonaphthyridine amines, les imidazotétrahydronaphthyridine amines, les oxazoloquinoline amines, les thiazoloquinoline amines, les oxazolopyridine amines, les thiazolopyridine amines, les oxazolonaphthyridine amines, les thiazolonaphthyridine amines, les pyrazolopyridine amines, les pyrazoloquinoline amines, les tétrahydropyrazoloquinoline amines, les pyrazolonaphthyridine amines, les tétrahydropyrazolonaphthyridine amines et les lH-imidazo dimères fusionnés en pyridine amines, quinoline amines, tétrahydroquinoline amines, naphthyridine amines ou tétrahydronaphthyridine amines. L'invention concerne également des procédés d'utilisation et des trousses.

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