C - Chemistry – Metallurgy – 07 – D
Patent
C - Chemistry, Metallurgy
07
D
167/228, 260/295
C07D 213/04 (2006.01) A61K 31/44 (2006.01) C07D 213/38 (2006.01) C07D 213/61 (2006.01) C07D 213/64 (2006.01) C07D 213/65 (2006.01) C07D 213/73 (2006.01) C07D 213/80 (2006.01) C07D 401/12 (2006.01)
Patent
CA 2008439
Abstract New aryl- and heteroarylethanol-pyridylalkylamines of the formula I Image (I) in which A represents =CH- or =N-, R0 represents hydrogen or methyl, R1 represents hydrogen, hydroxyl, halogen, cyano, alkyl, halogenoalkyl, hydroxyalkyl, alkoxy- carbonyl, aminocarbonyl, mono- and dialkylamino- carbonyl, alkoxy, halogenoalkoxy, halogenoalkyl- thio, NHSO2-alkyl, R2 represents hydrogen, hydroxyl, alkoxy or the radical -NR5R6, R3 represents the radicals specified for R1, R4 represents hydrogen, C1-C10-alkyl which is option- ally substituted by hydroxyl, halogen, alkoxy, acyloxy or radical -NR7R5, and represents the radical COR9 or the radical -O-Z-R10, Z represents C1-C10-alkylene, C2-C10-alkenylene or alkynylene, R3 represents hydrogen or alkyl, R6 represents hydrogen, alkyl, halogenoalkyl or acyl, it being possible for R5 and R6 to form, together with the adjoining N atom, a saturated or unsaturated heterocyclic 4-, 5- or 6-membered ring, R7 represents hydrogen optionally substituted alkyl, optionally substituted aryl, R8 represents the radicals specified for R7, R9 represents hydroxyl, alkoxy or the radical -NR7R8, R10 represents hydroxyl, alkoxy, acyloxy, optionally subtituted aryloxy or aralkyloxy, with the substituted R4 and the alkylamino group in the pryridyl ring of the formula I being in the p position with respect to one another or a physiologically tolerated salt therof, or, if A represents nitrogen, optionally the N-oxide thereof.
Berschauer Friedrich
Greife Heinrich A.
Hallenbach Werner
Klotz Gernot
Lindel Hans
Aktiengesellschaft Bayer
Berschauer Friedrich
Fetherstonhaugh & Co.
Greife Heinrich A.
Hallenbach Werner
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