Arylacrylamide derivatives

Details Arylacrylamide derivatives Arylacrylamide derivatives

C - Chemistry, Metallurgy

07

D

C07D 295/155 (2006.01) A61K 31/16 (2006.01) A61K 31/275 (2006.01) A61K 31/33 (2006.01) C07C 237/20 (2006.01) C07C 255/60 (2006.01) C07C 317/32 (2006.01) C07C 323/41 (2006.01) C07D 207/09 (2006.01) C07D 211/34 (2006.01) C07D 211/70 (2006.01) C07D 223/04 (2006.01) C07D 401/00 (2006.01) C07D 403/00 (2006.01) C07D 405/00 (2006.01) C07D 409/00 (2006.01) C07D 413/00 (2006.01) C07D 417/00 (2006.01)

Patent

CA 2206122

Compounds of the formula (See Fig.I) are useful psychotherapeutics and are potent serotonin (5-HT1) agonists and antagonists. Preferably, R1 is 4-methylpiper- azinyl, R2 is H, R3 is H or phenyl, R4 is phenyl, 3,4-dichloro- phenyl, 4-chlorobenzyl or 4-trichloromethylphenyl, R5 is H and X is H.

Les composés de formule (Voir Fig.I) sont utiles comme agents psychothérapeutiques et sont des agonistes et antagonistes puissants de la sérotonine (5-HT1). De préférence, R1 correspond à du 4-méthylpipérazinyle, R2 est H, R3 est H ou un phényle, R4 correspond à un phényle, à du 3,4-dichloro-phényle, à du 4-chlorobenzyle ou à du 4-trichlorométhylphényle, R5 est H et X est H.

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