C - Chemistry – Metallurgy – 07 – D
Patent
C - Chemistry, Metallurgy
07
D
C07D 403/06 (2006.01) A61K 31/41 (2006.01) A61K 31/44 (2006.01) A61K 31/505 (2006.01) A61K 31/675 (2006.01) C07D 233/70 (2006.01) C07D 249/12 (2006.01) C07D 401/14 (2006.01) C07D 403/10 (2006.01) C07D 403/14 (2006.01) C07D 405/14 (2006.01) C07D 409/14 (2006.01) C07F 9/645 (2006.01) C07F 9/6518 (2006.01)
Patent
CA 2050769
4-18240/A Azacyclic compounds Abstract Azacyclic compounds of the formula Image (I), wherein X is the group of the formula -C(R3)R4-[C(R5)R6]p-[C(R7)R8]q-(Ia) or the group of the formula -N(R9)-(Ib), R1 is unsubstituted or mono- or poly-substituted lower alkyl, lower alkenyl or lower alkynyl, it being possible for the substituents to be selected from the group consisting of hydroxy and halogen; cycloalkyl, cycloalkenyl, phenyl-lower alkyl, phenyl-lower alkenyl or phenyl-lower alkynyl, R2 is carboxy, 1H-tetrazol-5-yl, SO3H, PO2H2, PO3H2 or haloalkanesulfonylamino, either R3, R4,R5, R6, R7 and R8, independently of one another, are hydrogen, unsubstituted or mono- or poly-substituted lower alkyl, lower alkenyl or lower alkynyl, it being possible for the substituents to be selected from the group consisting of halogen, free or etherified hydroxy, free or esterified or amidated carboxy and unsubstituted or substituted amino; free or esterified or amidated carboxy, cycloalkyl, cycloalkenyl, an aliphatic hydrocarbon radical interrupted by O, or an aromatic radical, or one of the three pairs of variables R3/R4, R5/R6 and R7/R8 is a divalent aliphatic hydrocarbon radical and the variables of the other two pairs, independently of one another, are as defined above, R9 is hydrogen or unsubstituted or mono- or poly-substituted lower alkyl, lower alkenyl or lower alkynyl, it being possible for the substituents to be selected from the group consisting of free or etherified hydroxy and free or esterified or amidated carboxy, the indices p and q, independently of one another, are 0 or 1 and the rings A and B, independently of one another, are unsubstituted or substituted, and, if appropriate, the tautomers thereof, in each case in free form or in the form of salts, can be prepared in a manner known per se and can be used, for example, as activeingredients in medicaments.
Fuhrer Walter
Herold Peter
Ostermayer Franz
Ag Ciba-Geigy
Fetherstonhaugh & Co.
Fuhrer Walter
Herold Peter
Ostermayer Franz
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