Basic non-peptide bradykinin antagonists and pharmaceutical...

Details Basic non-peptide bradykinin antagonists and pharmaceutical... Basic non-peptide bradykinin antagonists and pharmaceutical...

C - Chemistry, Metallurgy

07

D

C07D 401/14 (2006.01) A61K 31/47 (2006.01) A61K 31/496 (2006.01) A61P 29/00 (2006.01) C07D 215/26 (2006.01) C07D 401/12 (2006.01)

Patent

CA 2488565

Non-peptide compounds of formula (I) having activity as specific antagonists of bradykinin (BK) B2 receptor. The compounds are chemically characterized by the presence of an alpha, alpha-disubstituted amino acid at least one amino group, free or salified, or the corresponding ammonium quaternary salt. These BK receptor antagonists are a novel class of medicaments which can be used in all the disorders in which said receptors are involved.

L'invention concerne des composés non peptidiques de formule (I) agissant comme des antagonistes spécifiques du récepteur B2 de bradykynine (BK). Lesdits composés se caractérisent sur le plan chimique par la présence d'un acide aminé alpha,alpha-disubstitué, au moins un groupe amino, libre ou salifié ou le sel quaternaire d'ammonium correspondant. Ces antagonistes du récepteur de BK constituent une nouvelle classe de médicaments pouvant s'utiliser dans tous les troubles où lesdits récepteurs sont impliqués.

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