Benzazine compounds and pharmaceutical uses thereof

Details Benzazine compounds and pharmaceutical uses thereof Benzazine compounds and pharmaceutical uses thereof

C - Chemistry, Metallurgy

07

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C07D 413/06 (2006.01) A61K 31/535 (2006.01) A61K 31/54 (2006.01) C07D 265/36 (2006.01) C07D 279/16 (2006.01) C07D 413/12 (2006.01) C07D 417/06 (2006.01) C07D 417/12 (2006.01) C07D 451/04 (2006.01) C07D 451/14 (2006.01) C07D 453/02 (2006.01)

Patent

CA 2020315

ABSTRACT OF THE DISCLOSURE A benzazine compound, a geometrical isomer of said benzazine compound, an optical isomer of said benzazine compound, and a pharmaceutically acceptable salt of said benzazine compound, said benzazine compound being represented by formula (I): Image wherein each symbol is as defined in the specification. Said benzazine compounds exhibit 5-HT3 receptor antagonistic activity, and 5-HT1A receptor and/or dopamine D2 receptor blocking activity so that they are useful as drugs for the prophylaxis or treatment of various digestive diseases vomiting and disturbances in central nervous systems and the like. The intermediates for said benzazine compounds are also disclosed.

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