Benzdioxane piperazine derivatives with a combination of...

Details Benzdioxane piperazine derivatives with a combination of... Benzdioxane piperazine derivatives with a combination of...

C - Chemistry, Metallurgy

07

D

C07D 405/12 (2006.01) A61K 31/496 (2006.01) A61P 25/00 (2006.01)

Patent

CA 2587940

The present invention relates to a group of novel 3 -(2-piperidin-4-yl-ethyl)- 1H-indole derivatives with a dual mode of action: serotonin reuptake inhibition and affinity for dopamine-D2 receptors and to methods for the preparation of these compounds. The invention also relates to the use of a compound disclosed herein for the manufacture of a medicament giving a beneficial effect. The compounds have the general formula (1) wherein the symbols have the meanings given in the specification.

L'invention concerne un groupe de nouveaux dérivés de 3 -(2-pipéridin-4-yl-éthyl)-1H-indole présentant un double mode d'action, à savoir une inhibition du recaptage de la sérotonine et une affinité pour les récepteurs de la dopamine-D2, ainsi que des procédés de préparation de ces composés. L'invention concerne également l'utilisation d'un desdits composés pour la préparation d'un médicament produisant un effet bénéfique. Les composés de l'invention sont représentés par la formule générale (1) dans laquelle les symboles ont la signification indiquée dans la description.

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