Benzenesulfonate salts of 4-fluoro-2-cyanopyrrolidine...

Details Benzenesulfonate salts of 4-fluoro-2-cyanopyrrolidine... Benzenesulfonate salts of 4-fluoro-2-cyanopyrrolidine...

C - Chemistry, Metallurgy

07

D

C07D 207/16 (2006.01) A61K 31/40 (2006.01) A61P 3/04 (2006.01) A61P 3/10 (2006.01) A61P 13/08 (2006.01) A61P 19/02 (2006.01) A61P 19/10 (2006.01) A61P 37/00 (2006.01) A61P 43/00 (2006.01)

Patent

CA 2496623

A benzenesulfonate salt of (2S,4S)-2-cyano-4-fluoro- 1-[(2-hydroxy-1,1-dimethyl)ethylamino]acetylpyrrolidine that has an excellent DPPIV inhibition activity as well as physical properties (e.g., stability) required for pharmaceutical preparations. The present invention allows easy obtaining of the compound in high-purity uniform crystal form with excellent solid-state stability.

La présente invention concerne un benzènesulfonate de (2S,4S)-2-cyano-4-fluoro-1-[(2-hydroxy-1,1-diméthyl)éthylamino]acétylpyrrolidine qui possède une excellente activité inhibitrice de la DPPIV et qui possède des propriétés souhaitables pour un médicament, telles qu'une stabilité élevée. Le composé de l'invention peut facilement être obtenu sous la forme de cristaux de stabilité élevée et de forme régulière, et il possède une stabilité élevée à l'état solide.

Affiliated with

Also associated with

Rating

Benzenesulfonate salts of 4-fluoro-2-cyanopyrrolidine... does not yet have a rating. At this time, there are no reviews or comments for this patent.

If you have personal experience with Benzenesulfonate salts of 4-fluoro-2-cyanopyrrolidine..., we encourage you to share that experience with our LandOfFree.com community. Your opinion is very important and Benzenesulfonate salts of 4-fluoro-2-cyanopyrrolidine... will most certainly appreciate the feedback.

Rate now

Comments { 0 }

Profile ID: LFCA-PAI-O-1838400