Benzodiazepine derivatives

Details Benzodiazepine derivatives Benzodiazepine derivatives

C - Chemistry, Metallurgy

07

D

C07D 401/04 (2006.01) A61K 31/55 (2006.01) A61K 31/69 (2006.01) C07D 401/14 (2006.01) C07D 403/04 (2006.01) C07D 403/14 (2006.01) C07D 405/14 (2006.01) C07D 417/14 (2006.01) C07D 453/00 (2006.01) C07D 471/08 (2006.01) C07D 487/08 (2006.01) C07F 5/02 (2006.01)

Patent

CA 2140008

Compounds of formula (I), and salts and prodrugs thereof, wherein R1 represents H, optionally substituted C1-6alkyl or C3-7cycloalkyl; R2 optionally substituted phenyl or R2 represents a group (A) where W is CH2 or NR10, and W1 is CH2, or W and W1 each represent O; R3 is C1-6alkyl, halo or NR13R14; R4 is H, C1-4alkyl, optionally substituted phenyl or optional- ly substituted benzyl; R5, R6, R7 and R8 are H or C1-4alkyl; or any two of R4, R5, R6, R7 and R8 together form a chain (CH2)t, and any other two of R4, R5, R6, R7 and R8 optionally form a chain (CH2)s where s and t are independently 1, 2 or 3; m is 2, 3, 4, 5, 6, 7, 8 or 9; n is 0, 1, 2, 3 or 4; and x is 0, 1, 2 or 3; are CCK and/or gastrin antagonists useful in therapy.

Affiliated with

Also associated with

Rating

Benzodiazepine derivatives does not yet have a rating. At this time, there are no reviews or comments for this patent.

If you have personal experience with Benzodiazepine derivatives, we encourage you to share that experience with our LandOfFree.com community. Your opinion is very important and Benzodiazepine derivatives will most certainly appreciate the feedback.

Rate now

Comments { 0 }

Profile ID: LFCA-PAI-O-1629422