C - Chemistry – Metallurgy – 07 – D
Patent
C - Chemistry, Metallurgy
07
D
C07D 405/12 (2006.01) A61K 31/40 (2006.01) A61P 25/18 (2006.01)
Patent
CA 2515541
The invention relates to novel benzofurane derivatives of formula (I) wherein R1, R2, X, Y, Z and m have the designations cited in patent claim 1. Said compounds have a strong affinity towards 5-HT1A receptors, inhibit the resumption of serotonin, have serotonin-agonistic and serotonin-antagonistic characteristics, and are suitable for using as antidepressants, anxiolytics, antipsychotics, neuroleptics and/or antihypertonics.
L'invention concerne de nouveaux dérivés de benzofurane de formule (I) dans laquelle R?1¿, R?2¿, X, Y, Z et m sont tels que définis dans la première revendication. Ces composés présentent une affinité élevée envers les récepteurs 5-HT¿1A?, empêchent la recapture de la sérotonine, constituent des agonistes et des antagonistes de la sérotonine et peuvent être utilisés en tant qu'antidépresseurs, anxiolytiques, antipsychotiques, neuroleptiques et/ou hypotenseurs.
Bartoszyk Gerd
Boettcher Henning
Heinrich Timo
Hoelzemann Guenter
Leibrock Joachim
Fetherstonhaugh & Co.
Merck Patent Gesellschaft Mit Beschraenkter Haftung
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