Benzoxazocines and their use as monoamine-reuptake inhibitors

Details Benzoxazocines and their use as monoamine-reuptake inhibitors Benzoxazocines and their use as monoamine-reuptake inhibitors

C - Chemistry, Metallurgy

07

D

C07D 267/22 (2006.01) A61K 31/395 (2006.01) A61K 31/422 (2006.01) A61P 29/00 (2006.01) C07D 221/00 (2006.01) C07D 267/00 (2006.01) C07D 413/04 (2006.01) C07D 498/04 (2006.01)

Patent

CA 2503172

Compounds of the general formula (1), wherein one of W, X, Y and Z is N or CR4 and the others are each CH; and R4 is a specified substituent. These compounds inhibit monoamine reuptake, and are useful in the treatment of pain, emesis depression, post traumatic stress disorders, attention deficit disorders, obsessive compulsive disorders, pre-menstrual syndrome, substance abuse and sexual dysfunction.

L'invention concerne des composés représentés par la formule générale (1), dans laquelle un membre de W, X, Y et Z représente N ou CR4, et les autres représentent chacun CH; et R4 représente un substituant déterminé. Ces composés inhibent la recapture des mono-amines, et sont efficaces pour le traitement de la douleur, des vomissements, de la dépression, des états de stress post-traumatiques, des troubles déficitaires de l'attention, des troubles obsessionnels compulsifs, du syndrome prémenstruel, des toxicomanies et des dysfonctions sexuelles.

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