C - Chemistry – Metallurgy – 07 – D
Patent
C - Chemistry, Metallurgy
07
D
C07D 295/088 (2006.01) A61K 31/16 (2006.01) A61K 31/404 (2006.01) A61K 31/4184 (2006.01) A61K 31/4465 (2006.01) A61K 31/4468 (2006.01) C07C 211/46 (2006.01) C07C 235/80 (2006.01) C07D 209/40 (2006.01) C07D 211/48 (2006.01) C07D 211/52 (2006.01) C07D 211/58 (2006.01) C07D 263/56 (2006.01)
Patent
CA 2552907
The invention relates to .beta.-ketoamide compounds of general formula (I) wherein the groups and radicals A, B, b, X, Y, Z, R1, R2, R3, R5a and R5b have the designations cited in patent claim 1. The invention also relates to medicaments containing at least one inventive amide. As a result of the MCH receptor antagonistic activity, the inventive medicaments are suitable for treating metabolic disorders and/or eating disorders, especially adipositas, bulimia, anorexia, hyperphagia and diabetes.
L'invention concerne des composés de cétoamides B de formule (I), dans laquelle les groupes et les restes A, B, b, X, Y, Z, R?1¿, R?2¿, R?3¿, R?5a¿ et R?5b¿ sont spécifiés dans la revendication 1. L'invention concerne, de plus, des médicaments comprenant au moins un amide de l'invention. Les médicaments de l'invention conviennent pour le traitement de troubles du métabolisme et/ou des troubles de l'appétit, en particulier l'adiposité, la boulimie, l'anorexie, l'hyperphagie et le diabète, grâce à l'activité antagoniste du récepteur de MCH.
Lehmann-Lintz Thorsten
Lotz Ralf Richard Hermann
Lustenberger Philipp
Mueller Stephan Georg
Roth Gerald-Juergen
Boehringer Ingelheim International Gmbh
Fetherstonhaugh & Co.
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