C - Chemistry – Metallurgy – 07 – C
Patent
C - Chemistry, Metallurgy
07
C
C07C 233/29 (2006.01) A61K 31/167 (2006.01) A61K 31/381 (2006.01) A61K 31/4164 (2006.01) A61K 31/4245 (2006.01) A61K 31/431 (2006.01) A61K 31/44 (2006.01) A61P 29/00 (2006.01) C07C 233/55 (2006.01) C07C 237/42 (2006.01) C07D 213/53 (2006.01) C07D 213/75 (2006.01) C07D 271/06 (2006.01) C07D 291/04 (2006.01) C07D 333/24 (2006.01) C07D 401/12 (2006.01)
Patent
CA 2602583
The invention is directed to novel vanilloid receptor type 1 (VR1) ligands. More specifically, the invention relates to novel biaryl-derived amides that are potent antagonists or agonists of VR1. Pharmaceutical and veterinary compositions and methods of treating mild to severe pain and various diseases using compounds of the invention are also described.
La présente invention a trait à de nouveaux ligands de récepteur vanilloïde de type 1 (VR1). De manière plus spécifique, l'invention a trait à de nouveaux amides dérivés de biaryle qui sont de puissants antagonistes ou agonistes de VR1. L'invention a également trait à des compositions pharmaceutiques et vétérinaires et à des procédés de traitement de douleur légère et sévère et de diverses maladies mettant en oeuvre les composés de l'invention.
Codd Ellen
Dax Scott L.
Flores Christopher
Jetter Michelle
Youngman Mark
Janssen Pharmaceutica N.v.
Ogilvy Renault Llp/s.e.n.c.r.l.,s.r.l.
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