Bicycloamine derivative

C - Chemistry – Metallurgy – 07 – D

Patent

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Details

C07D 451/06 (2006.01) A61K 31/439 (2006.01) A61K 31/46 (2006.01) A61K 31/4985 (2006.01) A61K 31/53 (2006.01) A61K 31/5377 (2006.01) A61K 31/5383 (2006.01) A61K 31/55 (2006.01) A61P 3/12 (2006.01) A61P 15/00 (2006.01) A61P 25/00 (2006.01) A61P 25/04 (2006.01) A61P 25/08 (2006.01) A61P 25/20 (2006.01) A61P 29/02 (2006.01) A61P 43/00 (2006.01) C07D 451/14 (2006.01) C07D 519/00 (2006.01)

Patent

CA 2714591

Compounds represented by formula (1) and pharmaceutically acceptable salts thereof have excellent sodium channel inhibitory action and are useful as therapeutic agents and analgesics for various kinds of neuralgia, neuropathy, epilepsy, insomnia, premature ejaculation and the like. (see formula I) wherein Q represents ethylene, etc., R1, R2 and R3 represent hydrogen, etc., X1 represents C1-6 alkylene, etc., X2 represents C1-6 alkylene, etc., A1 represents a 5- to 6-membered heterocyclic group, etc., and A2 represents C6-14 aryl, etc.

L'invention porte sur un composé représenté par la Formule (I) ou un sel pharmaceutiquement acceptable de celui-ci, qui a une excellente activité inhibitrice sur un canal sodique et est par conséquent utile comme agent thérapeutique pour divers types de névralgie, des troubles nerveux, l'épilepsie, l'insomnie, l'éjaculation précoce et autres ou comme agent analgésique. (I) où Q représente un éthylène ou similaire; R1, R2 et R3 représentent indépendamment un hydrogène ou similaire; X1 représente un alkylène en C1-6 ou similaire; X2 représente un alkylène en C1-6 ou similaire; A1 représente un groupe hétérocyclique à 5 à 6 chaînons ou similaire; et A2 représente un aryle en C6-14 ou similaire.

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